08/25/2007
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Diazepam (marketed under brand names Valium®, Stesolid®, Seduxen® and Apozepam®)
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anxiolytic, anticonvulsant, sedative, skeletal muscle relaxant and
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anxiety, insomnia, muscle spasms and some forms of epilepsy. Diazepam
is also used before certain medical procedures (such as endoscopies) to
reduce tension and anxiety, and in some surgical procedures to induce
amnesia.
Diazepam is a core medicine in the World Health Organization's
"Essential Drugs List", which is a list of minimum medical needs for a
basic health care system. Diazepam is used to treat a wide range of
conditions and is one of the most frequently prescribed benzodiazepines.
Diazepam was the second benzodiazepine to be invented by Leo Sternbach,
and was approved for use in 1963. Diazepam is five times more potent
than its predecessor, chlordiazepoxide, which it quickly surpassed in
terms of sales. After this initial success, other pharmaceutical
companies began to introduce other benzodiazepine derivatives.
The benzodiazepines gained popularity among medical professionals as an
improvement upon barbiturates, which have a comparatively narrow
therapeutic index, and are far more sedating at therapeutic doses. The
benzodiazepines are also far less dangerous; death rarely results from
diazepam overdose, except in cases where it is consumed with large
amounts of other depressants (such as alcohol or other sedatives).
Diazepam was the top-selling pharmaceutical in the United States from
1969 to 1982, with peak sales in 1978 of 2.3 billion pills.
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Over the years, physicians, psychiatrists and neurologists have
discovered many new off-label uses for diazepam, such as treatment of
spastic paresis and palliative treatment of stiff-person syndrome.
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